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Sinemet is a combination of carbidopa and levodopa applied in treatment of Parkinson's disease and Dopa-Responsive Dystonia. It prevents hypokinesia, stiffness, tremor, dysphagia, salivary discharge. Levodopa converts into dopamine owing to DOPA decarboxylase enzyme. Activation of central dopamine receptors improves the symptoms of Parkinson's disease and combination of carbidora reduces the unwanted peripheral side-effects of levodopa. Carbidopa usage increases the quantity of levodopa in the bloodstream that is available to enter the brain.
Sinemet (Levodopa/Carbidopa) Levodopa (also called L-dopa) is the most commonly prescribed and most effective drug for controlling the symptoms of Parkinson's disease, particularly bradykinesia and rigidity. Levodopa is transported to the nerve cells in the brain that produce dopamine.
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When carbidopa and levodopa are administered together, the half-life of levodopa is increased to about 1.5 hours. At steady state, the bioavailability of carbidopa from SINEMET tablets is approximately 99% relative to the concomitant administration of carbidopa and levodopa.
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